Binimetinib

Brand Name

Mektovi159,160,#

Pharmacology

Antineoplastic, mitogen-activated protein kinase 1 and 2 inhibitor

FDA Indication

BRAF-positive (V600E or V600K)d metastatic melanoma (in combination with encorafenib)

Similars

Cobimetinib, trametinib

Further Reading in Goodman & Gilman’s